a2b receptor antagonist — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T10058	A2B receptor antagonist 1		Adenosine Receptor
	A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.		Adenosine Receptor
T77508	A2B receptor antagonist 2 hydrochloride
	A2B receptor antagonist 2 hydrochloride is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T37793	A2B receptor antagonist 2	A2B receptor antagonist 2	Adenosine Receptor
	A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).		Adenosine Receptor
T21389	Enprofylline	Enprofilina,3-propylxanthine,3-n-Propylxanthine,Enprofyllinum	Others
	Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of sick...		Others
T23201	PSB 1115		Adenosine Receptor
	human A2B adenosine receptor antagonist		Adenosine Receptor
T27800	LAS38096	LAS 38096,LAS-38096	Adenosine Receptor
	LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .		Adenosine Receptor
T15715	LAS101057		Adenosine Receptor
	LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.		Adenosine Receptor
T27629	ISAM-140	ISAM140	Adenosine Receptor
	ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.		Adenosine Receptor
T23203	PSB-603	PSB 603	Adenosine Receptor
	PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.		Adenosine Receptor
T8512	BAY-545		Adenosine Receptor
	BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).		Adenosine Receptor
T15418	GS-6201	CVT-6883	Adenosine Receptor
	GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a Ki of 22 nM.		Adenosine Receptor
T16140	MRS 1754		Adenosine Receptor
	MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.		Adenosine Receptor
T22234	Alloxazine		Adenosine Receptor
	Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.		Adenosine Receptor
T14944	CGS 15943		PI3K , Adenosine Receptor
	CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM , respectively.		PI3K , Adenosine Receptor
T23197	PSB 0788		Others
	adenosine A2B receptor antagonist		Others
T26681	ATL802	ATL 802,ATL-802
	ATL802 is an adenosine A2B Receptor antagonist.
T26680	ATL-801
	ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.
T62611	Adenosine receptor antagonist 2
	Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.
T69675	PSB-1901 free base
	PSB-1901 is a potent A2B Adenosine Receptor Antagonist with Picomolar Potency (Ki 0.0835 nM, KB 0.0598 nM, human A2BAR) with >10 000-fold selectivity versus all other AR subtypes. PSB-1901 was similarly potent and select...
T61850	Adenosine receptor inhibitor 1
	Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR). It exhibits exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >100...